LGD 4033, Ligandrol, 5MG

SKU:
CAY-9002046-5MG
$36.00

Description

LGD 4033, Ligandrol

LGD 4033 is an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that binds to the androgen receptor with a Ki value of 1 nM.1 In animal models, LGD 4033 displays robust selectivity for muscle versus prostate tissues, anabolic activity in the muscle, and anti-resorptive and anabolic activity in bone.1 LGD 4033 has been abused as a performance-enhancing drug and the identification of its in vitro metabolites has been described.2,3 This product is intended for research and forensic applications.

WARNING This product is not for human or veterinary use.

Technical Information
Formal Name
4-[(2R)-2-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]-1-pyrrolidinyl]-2-(trifluoromethyl)-benzonitrile
CAS Number
1165910-22-4
Molecular Formula
C14H12F6N2O
Formula Weight
338.3
Purity
≥98%
Formulation(Request formulation change)
A crystalline solid
Solubility(Learn about Variance in Solubility)
  • DMF: 25 mg/ml
  • DMSO: 10 mg/ml
  • Ethanol: 25 mg/ml
  • Ethanol:PBS (pH 7.2) (1:5): 0.16 mg/ml
λmax
224, 295 nm
SMILES
O[C@@H](C(F)(F)F)[C@@]1([H])CCCN1C2=CC(C(F)(F)F)=C(C#N)C=C2
InChi Code
InChI=1S/C14H12F6N2O/c15-13(16,17)10-6-9(4-3-8(10)7-21)22-5-1-2-11(22)12(23)14(18,19)20/h3-4,6,11-12,23H,1-2,5H2/t11-,12?/m1/s1
InChi Key
OPSIVAKKLQRWKC-JHJMLUEUSA-N
Shipping & Storage Information
Storage
-20°C
Shipping
Wet ice in continental US; may vary elsewhere
Stability
≥ 4 years