LGD 4033, Ligandrol, 5MG

    • Description

    LGD 4033, Ligandrol

    LGD 4033 is an orally bioavailable, nonsteroidal selective androgen receptor modulator (SARM) that binds to the androgen receptor with a Ki value of 1 nM.1 In animal models, LGD 4033 displays robust selectivity for muscle versus prostate tissues, anabolic activity in the muscle, and anti-resorptive and anabolic activity in bone.1 LGD 4033 has been abused as a performance-enhancing drug and the identification of its in vitro metabolites has been described.2,3 This product is intended for research and forensic applications.

    WARNING This product is not for human or veterinary use.

    Technical Information
    Formal Name
    4-[(2R)-2-[(1R)-2,2,2-trifluoro-1-hydroxyethyl]-1-pyrrolidinyl]-2-(trifluoromethyl)-benzonitrile
    CAS Number
    1165910-22-4
    Molecular Formula
    C14H12F6N2O
    Formula Weight
    338.3
    Purity
    ≥98%
    Formulation(Request formulation change)
    A crystalline solid
    Solubility(Learn about Variance in Solubility)
    • DMF: 25 mg/ml
    • DMSO: 10 mg/ml
    • Ethanol: 25 mg/ml
    • Ethanol:PBS (pH 7.2) (1:5): 0.16 mg/ml
    λmax
    224, 295 nm
    SMILES
    O[C@@H](C(F)(F)F)[C@@]1([H])CCCN1C2=CC(C(F)(F)F)=C(C#N)C=C2
    InChi Code
    InChI=1S/C14H12F6N2O/c15-13(16,17)10-6-9(4-3-8(10)7-21)22-5-1-2-11(22)12(23)14(18,19)20/h3-4,6,11-12,23H,1-2,5H2/t11-,12?/m1/s1
    InChi Key
    OPSIVAKKLQRWKC-JHJMLUEUSA-N
    Shipping & Storage Information
    Storage
    -20°C
    Shipping
    Wet ice in continental US; may vary elsewhere
    Stability
    ≥ 4 years